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Flash Poster Presentations
Flash Poster Presentation Session 1
| KOLOCOURIS |
Antonios |
UNIVERSITY OF ATHENS |
FP01 |
NOVEL PYRAZOLO[3,4-C]PYRIDINE ANTAGONISTS WITH NANOMOLAR AFFINITY FOR A1 / A3 ADENOSINE RECEPTORS: BINDING KINETICS AND EXPLORATION OF THEIR BINDING PROFILE USING MUTAGENESIS EXPERIMENTS, MD SIMULATIONS AND TI/MD CALCULATIONS |
| BHELA |
Irene Preet |
UNIVERSITY OF PIEMONTE |
FP02 |
A STRAIGHTFORWARD SYNTHESIS OF PROTACS THROUGH MULTICOMPONENT REACTIONS |
| BOURGEAIS |
Mathieu |
UNIVERSITY OF BORDEAUX |
FP03 |
BIFUNCTIONAL CHEMICAL TOOLS FOR THE TARGETED DEGRADATION OF FURIN |
| NOCE |
Beatrice |
UNIVERSITY OF ROME |
FP04 |
NOVEL PYRIDINE-BASED HYDROXAMATES AND 2'-AMINOANILIDES AS HISTONE DEACETYLASE INHIBITORS: BIOCHEMICAL PROFILE AND ANTICANCER ACTIVITY |
| GRECO |
Francesco Aleksy |
GOETHE UNIVERSITY FRANKFURT |
FP05 |
CHEMICAL EXPLORATION OF THE ORTHOSTERIC AND ALLOSTERIC POCKETS OF DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 5 (MAP2K5/MEK5) BY SMALL MOLECULES |
| HUANG |
Rong |
PURDUE UNIVERSITY |
FP06 |
RATIONAL DEVELOPMENT OF POTENT AND SPECIFIC INHIBITORS FOR METHYLTRANSFERASES |
| DRAKOPOULOS |
Antonios |
UNIVERSITY OF GOTHENBURG |
FP07 |
EXPLORING THE MODE OF ACTION, THERMODYNAMIC PROFILE AND NUCLEOPHILE SELECTIVITY OF LABELLING WARHEADS FOR BRUTON'S TYROSINE KINASE |
| LOI |
Elena |
UNIVERSITY OF LJUBLJANA |
FP08 |
THE QUEST FOR THE FIRST POTENT IN VIVO ACTING OGT INHIBITOR |
| PROJ |
Matic |
UNIVERSITY OF LJUBLJANA |
FP09 |
REDOX ACTIVE OR THIOL REACTIVE? OPTIMIZATION OF RAPID SCREENS TO IDENTIFY LESS EVIDENT NUISANCE COMPOUNDS |
| KHEMAISSA |
Sonia |
SORBONNE UNIVERSITY |
FP10 |
DESIGN AND INTERNALIZATION PROPERTIES OF CHIMERIC CPP-GAG BINDING PEPTIDES |
Flash Poster Presentation Session 2
| BERABEZ |
Rayan |
UNIVERSITY OF ORLEANS |
FP11 |
SYNTHESIS AND PRECLINICAL VALIDATION OF LIMKS INHIBITORS: PROMISING DRUGS FOR OSTEOSARCOMA TREATMENT? |
| PAPANASTASIOU |
Ioannis |
NATIONAL AND KAPODISTRIAN UNIVERSITY OF ATHENS |
FP12 |
AN OVERVIEW OF THE ANTITRYPANOSOMAL PROFILE OF ADAMANTANE SCAFFOLDS |
| RICCIO |
Alessandra |
UNIVERSITY OF PERUGIA |
FP13 |
BEYOND CONVENTIONAL ANTI-CANCER AGENTS IN IMMUNOTHERAPY: HOW A TUMOR MICROENVIRONMENT LIMITATION COULD BE TURNED INTO AN ADVANTAGE |
| ESPELAND |
Ludvik |
UNIVERSITY OF BERGEN |
FP14 |
TARGETING A PSEUDOMONAS AERUGINOSA beta-KETOACYL-(ACYL-CARRIER-PROTEIN) SYNTHASE WITH COVALENT INHIBITORS INSPIRED BY CERULENIN |
| GANTER |
Benedikt |
UNIVERSITY OF HAMBURG |
FP15 |
SYNTHESIS OF MODIFIED T-1106-5´-TRIPHOSPHATES AS POTENTIAL INHIBITOR OF THE SARS-COV-2 RDRP |
| MARTIN SERRANO ORTIZ |
Angela |
UNIVERSITY OF GRENOBLE-ALPES |
FP16 |
PRECLINICAL EVALUATION OF ANTIBODY RECRUITING GLYCODENDRIMERS (ARGs) FOR CANCER THERAPHY |
| ZOLLO |
Michael |
TU MUNICH |
FP17 |
NEW CHEMOPROTEOMIC TECHNOLOGIES AND CHEMICAL MODALITIES FOR ANTIBIOTIC DISCOVERY |
| BRAUN |
Maria |
SPECS |
FP18 |
DISCOVERY AND OPTIMIZATION OF NOVEL ANTI-INFECTIVES TARGETING ISPE USING PROTEIN-TEMPLATED SYNTHESIS |
| UGOLINI |
Alessandra |
ITALIAN INSTITUTE OF TECHNOLOGY |
FP19 |
BACTERICIDAL AUTOPHAGY INHIBITORS TO TREAT RECURRENT INFECTIONS AND CANCER |
| KOVACHKA |
Sandra |
UNIVERSITY OF CÔTE D'AZUR |
FP20 |
PANICEIN A HYDROQUINONE AND ANALOGS OVERCOME CHEMOTHERAPY RESISTANCE IN CANCER CELL |
Flash Poster Session 1 (FP01-FP10)
- FP01 KOLOCOURIS Antonios UNIVERSITY OF ATHENS
NOVEL PYRAZOLO[3,4-C]PYRIDINE ANTAGONISTS WITH NANOMOLAR AFFINITY FOR A1 / A3 ADENOSINE RECEPTORS: BINDING KINETICS AND EXPLORATION OF THEIR BINDING PROFILE USING MUTAGENESIS EXPERIMENTS, MD SIMULATIONS AND TI/MD CALCULATIONS
- FP02 BHELA Irene Preet UNIVERSITY OF PIEMONTE
A STRAIGHTFORWARD SYNTHESIS OF PROTACS THROUGH MULTICOMPONENT REACTIONS
- FP03 BOURGEAIS Mathieu UNIVERSITY OF BORDEAUX
BIFUNCTIONAL CHEMICAL TOOLS FOR THE TARGETED DEGRADATION OF FURIN
- FP04 NOCE Beatrice UNIVERSITY OF ROME
NOVEL PYRIDINE-BASED HYDROXAMATES AND 2'-AMINOANILIDES AS HISTONE DEACETYLASE INHIBITORS: BIOCHEMICAL PROFILE AND ANTICANCER ACTIVITY
- FP05 GRECO Francesco Aleksy GOETHE UNIVERSITY FRANKFURT
CHEMICAL EXPLORATION OF THE ORTHOSTERIC AND ALLOSTERIC POCKETS OF DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 5 (MAP2K5/MEK5) BY SMALL MOLECULES
- FP06 HUANG Rong PURDUE UNIVERSITY
RATIONAL DEVELOPMENT OF POTENT AND SPECIFIC INHIBITORS FOR METHYLTRANSFERASES
- FP07 DRAKOPOULOS Antonios UNIVERSITY OF GOTHENBURG
EXPLORING THE MODE OF ACTION, THERMODYNAMIC PROFILE AND NUCLEOPHILE SELECTIVITY OF LABELLING WARHEADS FOR BRUTON'S TYROSINE KINASE
- FP08 LOI Elena UNIVERSITY OF LJUBLJANA
THE QUEST FOR THE FIRST POTENT IN VIVO ACTING OGT INHIBITOR
- FP09 PROJ Matic UNIVERSITY OF LJUBLJANA
REDOX ACTIVE OR THIOL REACTIVE? OPTIMIZATION OF RAPID SCREENS TO IDENTIFY LESS EVIDENT NUISANCE COMPOUNDS
- FP10 KHEMAISSA Sonia SORBONNE UNIVERSITY
DESIGN AND INTERNALIZATION PROPERTIES OF CHIMERIC CPP-GAG BINDING PEPTIDES
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Flash Poster Session 2 (FP11-FP20)
- FP11 BERABEZ Rayan UNIVERSITY OF ORLEANS
SYNTHESIS AND PRECLINICAL VALIDATION OF LIMKS INHIBITORS: PROMISING DRUGS FOR OSTEOSARCOMA TREATMENT?
- FP12 PAPANASTASIOU Ioannis UNIVERSITY OF ATHENS
AN OVERVIEW OF THE ANTITRYPANOSOMAL PROFILE OF ADAMANTANE SCAFFOLDS
- FP13 RICCIO Alessandra UNIVERSITY OF PERUGIA
BEYOND CONVENTIONAL ANTI-CANCER AGENTS IN IMMUNOTHERAPY: HOW A TUMOR MICROENVIRONMENT LIMITATION COULD BE TURNED INTO AN ADVANTAGE
- FP14 ESPELAND Ludvik UNIVERSITY OF BERGEN
TARGETING A PSEUDOMONAS AERUGINOSA beta-KETOACYL-(ACYL-CARRIER-PROTEIN) SYNTHASE WITH COVALENT INHIBITORS INSPIRED BY CERULENIN
- FP15 GANTER Benedikt UNIVERSITY OF HAMBURG
SYNTHESIS OF MODIFIED T-1106-5´-TRIPHOSPHATES AS POTENTIAL INHIBITOR OF THE SARS-COV-2 RDRP
- FP16 MARTIN SERRANO ORTIZ Angela UNIVERSITY OF GRENOBLE-ALPES
PRECLINICAL EVALUATION OF ANTIBODY RECRUITING GLYCODENDRIMERS (ARGs) FOR CANCER THERAPHY
- FP17 ZOLLO Michael TU MUNICH
NEW CHEMOPROTEOMIC TECHNOLOGIES AND CHEMICAL MODALITIES FOR ANTIBIOTIC DISCOVERY
- FP18 BRAUN Maria SPECS
DISCOVERY AND OPTIMIZATION OF NOVEL ANTI-INFECTIVES TARGETING ISPE USING PROTEIN-TEMPLATED SYNTHESIS
- FP19 UGOLINI Alessandra ITALIAN INSTITUTE OF TECHNOLOGY
BACTERICIDAL AUTOPHAGY INHIBITORS TO TREAT RECURRENT INFECTIONS AND CANCER
- FP20 KOVACHKA Sandra UNIVERSITY OF CÔTE D'AZUR
PANICEIN A HYDROQUINONE AND ANALOGS OVERCOME CHEMOTHERAPY RESISTANCE IN CANCER CELL
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Flash Poster Session 3 (FP21-FP30)
- FP21 TARKHANOVA Olga CHEMSPACE
ULTRA-LARGE CHEMICAL SPACES: APPROACHES TO BUILD AND EXPLORE
- FP22 BARTOS Piia UNIVERSITY OF EASTERN FINLAND
THE DARK SIDE OF MOLECULAR DYNAMICS SIMULATIONS: RNA-PROTEIN COMPLEXES
- FP23 DEGOTTE Gilles UNIVERSITY OF GRENOBLE-ALPES
DEVELOPMENT OF ENCODED COMBINATORIAL CHEMISTRY FOR THE IDENTIFICATION OF SPECIFIC LIGANDS OF G-QUADRUPLEX DNA STRUCTURES
- FP24 COTMAN Andrej Emanuel UNIVERSITY OF LJUBLJANA
CHIRAL INDANS VIA DYNAMIC KINETIC RESOLUTION: THREE-DIMENSIONAL BUILDING BLOCKS AND NATURAL PRODUCTS
- FP25 DINH Le Vi MONASH UNIVERSITY
DEVELOPMENT OF CALCIUM-SENSING RECEPTOR AGO-POSITIVE ALLOSTERIC MODULATORS, AC265347 DERIVATIVES, FOR THE TREATMENT OF HYPERPARATHYROIDISM AND RELATED DISORDERS
- FP26 COLSON Eloïse UNIVERSITY OF BERNE
EXPANDING THE MEDICINAL CHEMISTRY SYNTHETIC TOOLBOX WITH A RADICAL [3+3]-ANNULATION TOWARDS TROPANE AND RELATED ALKALOID SKELETONS
- FP27 MATVIYUK Tatiana ENAMINE
UNEXPECTED ISOMERIZATION OF OXETANE-CARBOXYLIC ACIDS
- FP28 MORGAN Barry UNIVERSITY OF TEXAS
DOES DNA-ENCODED LIBRARY TECHNOLOGY PROVIDE "NOVELTY"?
- FP29 MAKARA Gergely CHEMPASS
AI-ASSISTED GENERATIVE DESIGN OF SYNTHETICALLY FEASIBLE CHEMICAL SPACE FOR LEAD OPTIMIZATION
- FP30 REP Valentina UNIVERSITY OF ZAGREB
NOVEL REVERSED AMIDINE BENZOTHIAZOLES: DESIGN, SYNTHESIS, ANTITRYPANOSOMAL ACTIVITY AND ADME PROFILING
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Flash Poster Session 4 (FP31-FP40)
- FP31 PALAFERRI Leonardo UZH
A RATIONAL AND SYSTEMATIC APPROACH TO PROTACS DEVELOPMENT: IDENTIFICATION OF CBP/EP300 DEGRADERS
- FP32 CALZAFERRI Francesco CNRS
NOVEL STRATEGIES TO STUDY DNA METHYLATION IN HAEMATOLOGICAL CANCERS
- FP33 MAPLE Hannah BIO-TECHNE
VALIDATING TARGETS FOR TARGETED PROTEIN DEGRADATION USING DTAG ? A COMPREHENSIVE WORKFLOW SOLUTION
- FP34 GRISEL Clément CNRS
DESIGN OF CHEMICAL PROBES DERIVED FROM SCHWEINFURTHINS TO HIJACK OSBP
- FP35 RAMOS LLORCA Alba UANTWERP
ACTIVITY-BASED PROBES TARGETING TRYPSIN-LIKE SERINE PROTEASES FOR TARGET AND BIOMARKER DISCOVERY
- FP36 CORNER Thomas UNIVERSITY OF OXFORD
STRUCTURE-GUIDED OPTIMISATION OF SMALL-MOLECULE INHIBITORS OF THE HUMAN 2-OXOGLUTARATE-DEPENDENT OXYGENASE FACTOR INHIBITING HYPOXIA-INDUCIBLE FACTOR
- FP37 CHIEW Beatrice UNIVERSITY OF NEWCASTLE
DESIGN IN THE DARK - ILLUMINATING THE DRUGGABILITY OF 53BP1 FOR BRCA-1 BREAST CANCER
- FP38 BORLANDELLI Valentina LEIDEN UNIVERSITY
CYCLITOLS AS COVALENT INHIBITORS AND ACTIVITY-BASED PROBES FOR ?-D-GLUCURONIDASE AGAINST METABOLIC DRUG REACTIVATION AND CANCER PROGRESSION
- FP39 VAN WIER Suzanne UNIVERSITY OF EAST ANGLIA
REMOVING CANCER'S IMMORTALITY: TARGETING TELOMERASE
- FP40 VINAGREIRO Carolina LEIBNIZ INSTITUTE
ACTIVATABLE LUMINESCENT LANTHANOID PROBES FOR THE DETECTION OF VIRAL AND BACTERIAL INFECTIONS
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Flash Poster Session 5 (FP41-FP50)
- FP41 PROVENZANI Riccardo UNIVERSITY OF HELSINKI
MEMBRANE MOLECULAR DYNAMICS-ADJUVATED DESIGN AND SYNTHESIS OF MULTISUBSTITUTED PYRIDINES AS NOVEL PKC-TARGETED AGONISTS
- FP42 ZWERGEL Clemens UNIVERSITY OF ROME LA SAPIENZA
NOVEL SELENIUM CONTAING COMPOUNDS AS A PROMISE IN CANCER THERAPY? ABCB1 EFFLUX PUMP MODULATING AGENTS WITH CYTOTOXIC AND ANTIPROLIFERATIVE ACTIONS IN RESISTANT T-LYMPHOMA
- FP43 SHCHEHOLEVA Iryna UNIVERSITY OF COTE D'AZUR
ONCOGENIC MICRORNA INHIBITION BY SMALL MOLECULES: FRAGMENT-BASED DE NOVO LIGAND DESIGN AND SYNTHESIS
- FP44 BOFFEY Helen ALBORADA DRUG DISCOVERY INSTITUTE
DEVELOPMENT OF SELECTIVE, BRAIN PENETRANT PHOSPHATIDYLINOSITOL 5-PHOSPHATE 4-KINASE GAMMA INHIBITORS WITH CONTRASTING BINDING MODES
- FP45 NOZAL GARCIA Vanesa CIB - CSIC
RESCUING MOTOR NEURON DEGENERATION USING NOVEL MLK3 MODULATORS
- FP46 KRAUPNER Nicolas UNIVERSITY OF LILLE
IDENTIFICATION AND HIT MODULATION OF INDOLE-BASED ACTIVATORS OF THE INSULIN DEGRADING ENZYME
- FP47 KEIFF Francois LEIBNIZ INSITUTE
MODULATION OF THE MEISENHEIMER COMPLEX METABOLISM OF ANTIMYCOBACTERIAL BENZOTHIAZINONES
- FP48 OTAVA Tomáš IOCB PRAGUE
DESIGN AND SYNTHESIS OF S-ADENOSYLHOMOCYSTEINE ANALOGUES AS NANOMOLAR INHIBITORS OF SARS-COV-2 NSP14 METHYLTRANSFERASE
- FP49 LAPHOOKHIEO Surat MAE FAH LUANG UNIVERSITY
ALPHA-GLUCOSIDASE INHIBITORY ACTIVITY OF COMPOUNDS ISOLATED FROM FOUR ANNONACEAE PLANTS: DASYMASCHALON DASYMASCHALUM, DESMOS COCHINCHINESNSIS, POLYALTHIA CINNAMOMEA, AND TRIVALVARIA MACROPHYLLA
- FP50 DROP Marcin JAGIELLONIAN UNIVERSITY
NOVEL 5-HT6R NEUTRAL ANTAGONISTS DERIVED FROM 2-ARYLPYRROLE: CONTRIBUTION OF AGONIST-ACTIVATED STATES OF THE RECEPTOR TO NEUROTOXICITY
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Flash Poster Session 6 (FP51-FP60)
- FP51 COLCHON-PIERNA Esther UNIVERSITY OF SANTIAGO DE COMPOSTELA
FREE LABELLING PLATFORM TO DETERMINE DRUG BINDING TO PROTEINS
- FP52 JOCH Melanie LEIBNIZ INSTITUTE
A CELL-BASED METABOLIC ASSAY FOR HYDRIDE MEISENHEIMER FORMATION ASSESSMENT TO GUIDE LEAD OPTIMIZATION OF NEXT-GENERATION ANTITUBERCULAR BENZOTHIAZINONES
- FP53 GENTILINI Emilie UNIVERSITY OF CÔTE D'AZUR
NOVEL METHODOLOGIES FOR THE SYNTHESIS OF POLYCYCLIC DERIVATIVES USING GOLD AND CARBOPHILIC METAL CATALYSIS
- FP54 POCHET Lionel UNAMUR
TOWARDS NEW FXIIa INHIBITORS BY APPLICATION OF A FRAGMENT-BASED LEAD DISCOVERY APPROACH AND AFFINITY CAPILLARY ELECTROPHORESIS SCREENING ASSAY
- FP55 NOWICKI Krzysztof WARSAW UNIVERSITY OF TECHNOLOGY
THE USE OF THIOL-FUNCTIONALIZED BENZOSILOXABOROLES FOR ACHIEVING DIVERSE SUBSTITUTION PATTERNS - BIOLOGICAL EVALUATION OF NOVEL PROMISING ANTIBACTERIAL AGENTS
- FP56 LEBERECHT Christoph PHARMAI
GENERATION OF FOCUSED LIBRARIES: AI-POWERED REDUCTION OF LARGE COMPOUND LIBRARIES LEADS TO THE DISCOVERY OF NOVEL INHIBITORS OF SIRTUIN-1
- FP57 MULLIRI Kleni UNIVERSITY OF BERN
SAR OF TRIQUINAZINE, A CLASS OF POTENT JANUS KINASE INHIBITORS
- FP58 TARDIA Piero CHARLES RIVER LABORATORIES
DISCOVERY OF A NOVEL CLASS OF D-AMINO ACID OXIDASE INHIBITORS USING THE SCHRÖDINGER COMPUTATIONAL PLATFORM
- FP59 SAN Carine CNAM
OPTIMIZATION OF A SYNTHETIC STEP USING A DESIGN OF EXPERIMENTS APPROACH: APPLICATION TO A LATE-STAGE RADIOLABELING METHOD BY ALUMINIUM-[18F]FLUORIDE COORDINATION
- FP60 SCHEIBELBERGER Lukas UNIVERSITY OF VIENNA
SYNTHESIS OF 4-DEOXY-4-FLUORO-D-SEDOHEPTULOSE AND AN APPROACH FOR ITS FLUORINE-18 LABELED ANALOGUE
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