| Sunday April 21, 2024 |
| 17:30 | Registration |
|
| 19:30 | Dinner at the Hotel |
|
| 21:00 | Get Together at the Castle Bar |
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| Monday April 22, 2024 |
| 07:15 | Breakfast |
|
| 08:15 | Opening Ceremony |
Prof. Laura HEITMAN
(UNIVERSITY OF LEIDEN, Leiden, The Netherlands) |
| 08:30 | Physicochemical Property Considerations in Modern Drug Discovery and Implications for Hit Finding and Library Design - Part 1 |
Prof. Mike WARING (NEWCASTLE UNIVERSITY, Newcastle upon Tyne, United Kingdom)
Dr Hannah STEWART (NEWCASTLE UNIVERSITY, Newcastle Upon Tyne, United Kingdom) |
| 10:00 | Coffee Break |
|
| 10:30 | Physicochemical Property Considerations in Modern Drug Discovery and Implications for Hit Finding and Library Design - Part 2 |
Prof. Mike WARING (NEWCASTLE UNIVERSITY, Newcastle upon Tyne, United Kingdom)
Dr Hannah STEWART (NEWCASTLE UNIVERSITY, Newcastle Upon Tyne, United Kingdom) |
| 12:00 | Lunch & Group Picture |
|
| 13:30 | What Can We Learn from 20+ years of Fragment Based Drug Discovery and What Are the Future Opportunities? - Part 1 |
Dr Christopher JOHNSON
(ASTEX PHARMACEUTICALS, Cambridge, United Kingdom) |
| 15:00 | Coffee Break |
|
| 15:30 | What Can We Learn from 20+ years of Fragment Based Drug Discovery and What Are the Future Opportunities? - Part 2 |
Dr Christopher JOHNSON
(ASTEX PHARMACEUTICALS, Cambridge, United Kingdom) |
| 17:00 | Day End |
|
| 18:00 | Walking tour through Leiden |
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| 19:30 | Dinner in Leiden |
|
| Tuesday April 23, 2024 |
| 08:30 | Enabling Drug Discovery Projects with Encoded Library Technologies - Part 1 |
Dr Frederic BERST (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Basel, Switzerland)
Dr Christoph DUMELIN (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Basel, Switzerland) |
| 10:00 | Coffee Break |
|
| 10:30 | Enabling Drug Discovery Projects with Encoded Library Technologies - Part 2 |
Dr Frederic BERST (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Basel, Switzerland)
Dr Christoph DUMELIN (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Basel, Switzerland) |
| 12:00 | Lunch |
|
| 13:30 | Design of Multifunctional Conjugates for the Targeting of Non-coding RNAs: Anticancer and Antimicrobial Applications |
Dr Maria DUCA
(UNIVERSITY OF CÔTE D'AZUR, Nice, France) |
| 15:00 | Coffee Break |
|
| 15:30 | Activity Based Profiling as Tool in Medicinal Chemistry |
Prof. Mario VAN DER STELT
(UNIVERSITY OF LEIDEN, Leiden, The Netherlands) |
| 17:00 | Day End |
|
| 19:30 | Dinner at the hotel |
|
| 21:00 | Get Together at the Castle Bar |
|
| Wednesday April 24, 2024 |
| 07:00 | Breakfast |
|
| 08:30 | General Considerations for Covalent Drug Discovery Exemplified with Acalabrutinib |
Dr Gerjan DE BRUIN
(ACERTA PHARMA, Oss, The Netherlands) |
| 10:00 | Coffee Break |
|
| 10:30 | Discovery of Zosurabalpin |
Dr Patrizio MATTEI
(ROCHE INNOVATION CENTER BASEL, Basel, Switzerland) |
| 12:00 | Wrap up and Lunch |
|
